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    Chiral Phosphoric Acid Catalyzed Oxidative Kinetic Resolution of Indolines Based on Transfer Hydrogenation to Imines

    Saito, K.; Shibata, Y.; Yamanaka, M.; Akiyama, T, J. Am. Chem. Soc. 2013, 135, 11740-11743.

    Hydrodefluorinations of Trifluorotoluenes by LiAlH4 and TiCl4

    Akiyama, T.; Atobe, K.; Shibata, M.; Mori, K. J. Fluorine Chem. 2013, 152, 81-83.

    Enantioselective Synthesis of Multisubstituted Biaryl Skeleton by Chiral Phosphoric Acid Catalyzed Desymmetrization/Kinetic Resolution Sequence

    Mori, K.; Ichikawa, Y.; Kobayashi, M.; Shibata, Y.; Yamanaka, M.; Akiyama, T. J. Am. Chem. Soc. 2013, 135 , 3964-3970.

    Molecular Iodine Catalyzed Transfer Hydrogenation: Reduction of Aldimines, Ketimines, and a-Imino esters

    Bachu, P.; Zhu, C.; Akiyama, T. Tetrahedron Lett. 2013, 54, 3977-3981.

    Kinetic Resolution in Chiral Bronsted Acid Catalyzed Aldol Reaction: Enantioselective Robinson-type Annulation Reaction

    Yamanaka, M.; Hoshino, M.; Katoh, T.; Mori, K.; Akiyama, T. Eur. J. Org. Chem. 2012, 4508-4514.

    Phopshoric Acid Catalyzed Enantioselective Transfer Deruteration of Ketimines by Use of Benzothiazoline as a Deuterium Donor: Synthesis of Optically Active Deuterated Amines

    Sakamoto, T.; Mori, K.; Akiyama, T. Org. Lett. 2012, 14, 3312-3315.

    Enantioselective Organocatalytic Reductive Amination of Aliphatic Ketones by Benzothiazoline as Hydrogen Donor

    Saito, K.; Akiyama, T. Chem. Commun. 2012, 48, 4573-4575.

    Concise Route to 3-Arylisoquinoline Skeleton by Lewis Acid Catalyzed C(sp3)-H Bond Functionalization and Its Application to Formal Synthesis of (+-)-Tetrahydropalmatine

    Mori, K.; Kawasaki, T.; Akiyama, T. Org. Lett. 2012, 14, 1436-1439.

    Carboxyl-Tailed Benzothiazoline: A Readily Removable Hydrogen Donor for the Transfer Hydrogenation of Imines

    Zhu, C.; Akiyama, T. Tetrahedron Lett. 2012, 53, 416-418.

    Rapid Access to 3-Aryltetraline Skeleton via C(sp3)-H Bond Functionalization: Investigation on the Substituent Effect of Aromatic Ring Adjacent to C-H Bond in Hydride Shift/Cyclization Sequence

    Mori, K.; Sueoka, S.; Akiyama, T. Chem. Lett. 2011, 40 , 1386-1388.

    Development of Chiral Bronsted Acid and its Application to Asymmetric Synthesis

    T. Akiyama, J. Synth. Org. Chem. Jpn., 2011, 69, 913-925.

    Chiral Phosphoric Acid Catalyzed Transfer Hydrogenation: A Facile Synthetic Access to Highly Optically Active Trifluoromehylated Amines

    Henseler, A.; Kato, M.; Mori, K.; Akiyama, T. Angew. Chem. Int. Ed. 2011, 50, 8180-8183.

    Bronsted Acid Catalyzed Reductive Amination with Benzothiazoline as a Hyighly Efficient Hydrogen Donor

    Zhu, C.; Akiyama, T. Synlett (Cluster, Bronsted Acid, invited), 2011, 1251-1254.

    Selective Activation of Enantiotopic C(sp3)-Hydrogen by Means of Chiral Phosphoric Acid: Asymmetric Synthesis of Tetrahydroquinoline Derivatives

    Mori, K.; Ehara, K.; Kurihara, K.; Akiyama, T. J. Am. Chem. Soc. 2011, 133, 6166-6169.

    Chiral Phosphoric Acid Catalyzed Enantioselective Synthesis of b-Amino-a,a-difluoro Carbonyl Compounds

    Kashikura, W.; Mori, K.; Akiyama, T. Org. Lett. 2011, 13, 1860-1863.