Concise Route to 3-Arylisoquinoline Skeleton by Lewis Acid Catalyzed C(sp3)-H Bond Functionalization and Its Application to Formal Synthesis of (+-)-Tetrahydropalmatine
Mori, K.; Kawasaki, T.; Akiyama, T. Org. Lett. 2012, 14, 1436-1439.
Carboxyl-Tailed Benzothiazoline: A Readily Removable Hydrogen Donor for the Transfer Hydrogenation of Imines
Rapid Access to 3-Aryltetraline Skeleton via C(sp3)-H Bond Functionalization: Investigation on the Substituent Effect of Aromatic Ring Adjacent to C-H Bond in Hydride Shift/Cyclization Sequence
Mori, K.; Sueoka, S.; Akiyama, T. Chem. Lett. 2011, 40 , 1386-1388.
Development of Chiral Bronsted Acid and its Application to Asymmetric Synthesis
Chiral Phosphoric Acid Catalyzed Transfer Hydrogenation: A Facile Synthetic Access to Highly Optically Active Trifluoromehylated Amines
Henseler, A.; Kato, M.; Mori, K.; Akiyama, T. Angew. Chem. Int. Ed. 2011, 50, 8180-8183.
Bronsted Acid Catalyzed Reductive Amination with Benzothiazoline as a Hyighly Efficient Hydrogen Donor
Zhu, C.; Akiyama, T. Synlett (Cluster, Bronsted Acid, invited), 2011, 1251-1254.
Selective Activation of Enantiotopic C(sp3)-Hydrogen by Means of Chiral Phosphoric Acid: Asymmetric Synthesis of Tetrahydroquinoline Derivatives
Mori, K.; Ehara, K.; Kurihara, K.; Akiyama, T. J. Am. Chem. Soc. 2011, 133, 6166-6169.
Chiral Phosphoric Acid Catalyzed Enantioselective Synthesis of b-Amino-a,a-difluoro Carbonyl Compounds
Kashikura, W.; Mori, K.; Akiyama, T. Org. Lett. 2011, 13, 1860-1863.
Expeditious Construction of a Carbobicyclic Skeleton via a sp3-C-H Functionalization: Hydride Shift from an Aliphatic Tertiary Position in an Internal Redox Process
Mori, K.; Sueoka, S.; Akiyama, T. J. Am. Chem. Soc. 2011, 133, 2424-2426.
Chiral Bronsted Acid-Catalyzed Asymmetric Friedel-Crafts Alkylation of Indoles with a,b-Unsaturated Ketones: Short Access to Optically Active 2- and 3-Substituted Indole Derivatives
Sakamoto, T.; Itoh, J.; Mori, K.; Akiyama, T. Org. Biomol. Chem. 2010, 8, 5448-5454.
A One-pot Tandem Approach of Synthesis of Benzothiazoles from Benzyl Halides
Benzothiazoline: Highly Efficient Reducing Agent for the Enantioselective Organocatalytic Transfer Hydrogenation of a-Imino Esters
Zhu, C.; Akiyama, T. Adv. Synth. Catal. 2010, 352, 1846-1850.
Niobium-catalyzed Activation of CF3 Group on Alkene: Synthesis of Substituted Indenes
Fuchibe, K.; Atobe, K.; Fujita, Y.; Mori, K.; Akiyama, T. Chem. Lett. 2010, 39, 867-869.
Synthesis and Properties of Phosphoroselenoic Acids, and their Salts Bearing Binaphthyl Groups
Murai, T.; Monzaki, M.; Katoh, T.; Suzuki, T.; Akiyama, T. Phosphorus, Sulfur, Silicon Relat. Elem. 2010, 185, 964-973.
Enantioselective Friedel-Crafts Alkylation Reaction of Indoles with a,b-Unsaturated Acyl Phosphonates Catalyzed by Chiral Phosphoric Acid